The novel formulation of silybin / ß-cyclodextrin inclusion complex makes silybin, the main active constituent of Silymarin, immediately bioavailable. Upon administration, an association-dissociation equilibrium is rapidly established with free individual silybin molecules readily available for absorption (in contrast to clumping which usually occurs with conventional tablet and capsule forms).

silybin / ß-cyclodextrin inclusion complex   ß-cyclodextrin molecule single silybin molecule

Single silybin melocules are instantaneously absorbed and the equilibrium is rapidly shifted to the right hand side.